Found 6 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50464180'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Vanderbilt Univercity
Curated by ChEMBL
Vanderbilt Univercity
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Positive allosteric modulation of human M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretrea...More data for this Ligand-Target Pair
Affinity DataEC50: 2.29E+3nMAssay Description:Agonist activity at rat M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye base...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Vanderbilt Univercity
Curated by ChEMBL
Vanderbilt Univercity
Curated by ChEMBL
Affinity DataEC50: 123nMAssay Description:Agonist activity at human M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye ba...More data for this Ligand-Target Pair
Affinity DataEC50: 95nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 2.29E+3nMAssay Description:Agonist activity at rat M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye base...More data for this Ligand-Target Pair