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Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50464189'
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Univercity

Curated by ChEMBL
LigandPNGBDBM50464189(CHEMBL4240041)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at rat M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye base...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Univercity

Curated by ChEMBL
LigandPNGBDBM50464189(CHEMBL4240041)
Affinity DataEC50:  1.21E+3nMAssay Description:Agonist activity at rat M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye base...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Univercity

Curated by ChEMBL
LigandPNGBDBM50464189(CHEMBL4240041)
Affinity DataEC50:  40nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Univercity

Curated by ChEMBL
LigandPNGBDBM50464189(CHEMBL4240041)
Affinity DataEC50:  42nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed