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Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50265994'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50265994(CHEMBL4068393)
Affinity DataKi:  0.710nMAssay Description:Displacement of [3H]NMS from human muscarinic acetylcholine receptor M2 expressed in CHOK9 cells after 3 hrs by liquid scintillation counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50265994(CHEMBL4068393)
Affinity DataKd:  8.40nMAssay Description:Binding affinity to human muscarinic acetylcholine receptor M2 expressed in live adherent CHOK9 cells after 2 hrs by liquid scintillation counting as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50265994(CHEMBL4068393)
Affinity DataKd:  3nMAssay Description:Binding affinity to human muscarinic acetylcholine receptor M2 expressed in CHOK9 cell homogenate after 2 hrs by liquid scintillation counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50265994(CHEMBL4068393)
Affinity DataKd:  4.60nMAssay Description:Binding affinity to human muscarinic acetylcholine receptor M2 expressed in CHOK9 cell homogenate assessed as ratio of dissociation rate constant to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed