Found 7 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50452855'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of W£Rzburg
Curated by ChEMBL
University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M2 receptor expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of W£Rzburg
Curated by ChEMBL
University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 W422A mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of W£Rzburg
Curated by ChEMBL
University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of W£Rzburg
Curated by ChEMBL
University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y177Q/T423H mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Binding affinity towards rat Muscarinic acetylcholine receptor M2 was determinedMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of W£Rzburg
Curated by ChEMBL
University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 Y104A mutant expressed in Flp-In-CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKd: 3nMAssay Description:In vitro receptor binding against Muscarinic acetylcholine receptor M2 in rat heart was determined using [3H]pirenzepineMore data for this Ligand-Target Pair