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Report error Found 3 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M3' and Ligand = 'BDBM50181089'
TargetMuscarinic acetylcholine receptor M3(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50181089(6-(azepan-1-yl)-N,2-dicyclopropyl-5-methylpyrimidi...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50181089(6-(azepan-1-yl)-N,2-dicyclopropyl-5-methylpyrimidi...)
Affinity DataKi:  3.20nMAssay Description:Antagonist activity at muscarinic M3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50181089(6-(azepan-1-yl)-N,2-dicyclopropyl-5-methylpyrimidi...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]N-methylscopolamine from human recombinant M3 muscarinic receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed