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Found 2 Enz. Inhib. hit(s) with Target = 'Neprilysin' and Ligand = 'BDBM153117'
TargetNeprilysin(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM153117(US8993631, 20 | US9006249, Example 9-1 | US9603819...)
Affinity DataIC50:  142nMAssay Description:The activity of a compound according to the present invention can be assessed by the following in vitro & in vivo methods and/or by the following in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNeprilysin(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM153117(US8993631, 20 | US9006249, Example 9-1 | US9603819...)
Affinity DataIC50:  142nMpH: 7.4 T: 2°CAssay Description:See A fluorescence lifetime-based assay for protease inhibitor profiling on human kallikrein 7 Doering K, Meder G, Hinnenberger M, Woelcke J, Mayr L ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent