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Report error Found 3 Enz. Inhib. hit(s) with Target = 'Neuromedin-K receptor' and Ligand = 'BDBM362850'
TargetNeuromedin-K receptor(Human)
Oged

US Patent
LigandPNGBDBM362850((R)-(8-methyl-3-(2- (trifluoromethyl)thiazol-4-yl)...)
Affinity DataKi:  29nMAssay Description:The ability of compounds of the invention to inhibit the binding of the NK-3 receptor selective antagonist 3H-SB222200 was assessed by an in vitro ra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetNeuromedin-K receptor(Human)
Oged

US Patent
LigandPNGBDBM362850((R)-(8-methyl-3-(2- (trifluoromethyl)thiazol-4-yl)...)
Affinity DataKi:  29nMAssay Description:The ability of compounds of the invention to inhibit the binding of the NK-3 receptor selective antagonist 3H-SB222200 was assessed by an in vitro ra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetNeuromedin-K receptor(Human)
Oged

US Patent
LigandPNGBDBM362850((R)-(8-methyl-3-(2- (trifluoromethyl)thiazol-4-yl)...)
Affinity DataIC50:  33nMAssay Description:The ability of compounds of the invention to inhibit the binding of the NK-3 receptor selective antagonist 3H-SB222200 was assessed by an in vitro ra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent