Report error Found 26 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4' and Ligand = 'BDBM50049757'
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 0.0100nMAssay Description:Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand bindi...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Human)
University of Bath
Curated by PDSP Ki Database
University of Bath
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Human)
University of Bath
Curated by PDSP Ki Database
University of Bath
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Human)
University of Bath
Curated by PDSP Ki Database
University of Bath
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 0.0350nMAssay Description:Displacement of [3H]nicotine from alpha4beta2 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 0.0470nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 0.0470nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Human)
University of Bath
Curated by PDSP Ki Database
University of Bath
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Human)
University of Bath
Curated by PDSP Ki Database
University of Bath
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 0.0610nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 0.0610nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Human)
University of Bath
Curated by PDSP Ki Database
University of Bath
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse
Curated by PDSP Ki Database
National Institute On Drug Abuse
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Human)
University of Bath
Curated by PDSP Ki Database
University of Bath
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Mouse)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 0.0370nMAssay Description:Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylc...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Human)
University of Bath
Curated by PDSP Ki Database
University of Bath
Curated by PDSP Ki Database
Affinity DataEC50: 120nMAssay Description:Agonist activity at human recombinant alpha4beta2 nAChR expressed in human IMR32 cells assessed as calcium dynamics by FLIPR assayMore data for this Ligand-Target Pair