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Found 2 Enz. Inhib. hit(s) with Target = 'Nociceptin receptor' and Ligand = 'BDBM50335573'
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50335573((1-{4-[2-(3,3-Dimethylpiperazin-1-yl)-1H-benzimida...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50335573((1-{4-[2-(3,3-Dimethylpiperazin-1-yl)-1H-benzimida...)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human NOP receptor expressed in HEK293 cells assessed as induction of [35S]GTPgammaS binding after 30 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed