Affinity DataIC50: 3.10nMAssay Description:Inverse agonist activity at human His6-tagged RORgammat LBD (264 to 518 residues) assessed as reduction in biotinylated RIP140 co-activator recruitme...More data for this Ligand-Target Pair
Affinity DataKd: 465nMAssay Description:Binding affinity to RORgammat (unknown origin) by reporter displacement assayMore data for this Ligand-Target Pair
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