Found 3 Enz. Inhib. hit(s) with Target = 'Orexin/Hypocretin receptor type 1' and Ligand = 'BDBM50028059'
Affinity DataKi: 1.58E+3nMAssay Description:Binding affinity to human OX1 receptor expressed in CHO cell membranes by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+3nMAssay Description:Binding affinity to human orexin-1 receptor expressed in CHO cell membranes after 3 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.79E+3nMAssay Description:Antagonist activity at human OX1R expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair