Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Orexin/Hypocretin receptor type 1' and Ligand = 'BDBM50028059'
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50028059(CHEMBL3338866)
Affinity DataKi:  1.58E+3nMAssay Description:Binding affinity to human OX1 receptor expressed in CHO cell membranes by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50028059(CHEMBL3338866)
Affinity DataKi:  1.58E+3nMAssay Description:Binding affinity to human orexin-1 receptor expressed in CHO cell membranes after 3 hrs by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50028059(CHEMBL3338866)
Affinity DataIC50:  1.79E+3nMAssay Description:Antagonist activity at human OX1R expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed