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Found 3 Enz. Inhib. hit(s) with Target = 'Orexin receptor type 2' and Ligand = 'BDBM50092810'
TargetOrexin receptor type 2(Homo sapiens (Human))TBA
LigandPNGBDBM50092810(CHEMBL3586412)
Affinity DataKi:  5nMAssay Description:Antagonist activity at human OX2R by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOrexin receptor type 2(Homo sapiens (Human))TBA
LigandPNGBDBM50092810(CHEMBL3586412)
Affinity DataKi:  25nMAssay Description:Displacement of (S)-N-(2-(1H-pyrrol-1-yl)phenyl)-1-(2-((3H)-1-methyl-1H-benzo[d]imidazol-2-ylthio)acetyl)pyrrolidine-2-carboxamide from human OX2 rec...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))TBA
LigandPNGBDBM50092810(CHEMBL3586412)
Affinity DataIC50:  98nMAssay Description:Antagonist activity at OX2R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed