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Report error Found 6 Enz. Inhib. hit(s) with Target = 'P2X purinoceptor 4' and Ligand = 'BDBM50506158'
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50:  108nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Mouse)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50:  112nMAssay Description:Antagonist activity at mouse P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50:  211nMAssay Description:Antagonist activity at human P2X4 receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50:  211nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Rat)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50:  233nMAssay Description:Antagonist activity at rat P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50:  320nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of inhibition of ATP-evoked current at -90 mV hold...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed