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Found 3 Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 12' and Ligand = 'BDBM50298159'
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50298159((4S)5-Oxo-5-{4-[(pentyloxy)carbonyl]piperazin-1-yl...)
Affinity DataKi:  11nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50298159((4S)5-Oxo-5-{4-[(pentyloxy)carbonyl]piperazin-1-yl...)
Affinity DataKi:  11nMAssay Description:Displacement of [33P]ADP from human recombinant P2Y12 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50298159((4S)5-Oxo-5-{4-[(pentyloxy)carbonyl]piperazin-1-yl...)
Affinity DataIC50:  1.50E+4nMAssay Description:Antagonist activity at human P2Y12 receptor assessed as inhibition of ADP-induced platelet-rich plasma aggregation by turbidimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed