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Found 2 Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 12' and Ligand = 'BDBM50298184'
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50298184((S)-4-(4-(benzyloxy)-6-phenylpicolinamido)-5-(4-(e...)
Affinity DataKi:  28nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50298184((S)-4-(4-(benzyloxy)-6-phenylpicolinamido)-5-(4-(e...)
Affinity DataIC50:  3.10E+4nMAssay Description:Antagonist activity at human P2Y12 receptor assessed as inhibition of ADP-induced platelet-rich plasma aggregation by turbidimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed