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TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences
Curated by ChEMBL
Inception Sciences
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Antagonist activity at human PPAR-alpha assessed as inhibition of GW7647-induced effect after overnight incubation by cell-based luciferase reporter ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences
Curated by ChEMBL
Inception Sciences
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:Antagonist activity at GST-tagged PPAR-alpha (unknown origin) assessed as inhibition of GW7647-induced effect after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences
Curated by ChEMBL
Inception Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPAR-alphaMore data for this Ligand-Target Pair
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