Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM29887'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Amgen

LigandPNGBDBM29887(alkynyl ether, 29)
Affinity DataKi:  30nM EC50:  300nMAssay Description:The human PPARgamma ligand binding was directly measured using a filtration assay in a UniFilter 350 96-well assay plate (Polyfiltronics). The reacti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed