Found 3 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50389161'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College
Curated by ChEMBL
Trinity College
Curated by ChEMBL
Affinity DataEC50: 5.45E+3nMAssay Description:Binding affinity to PPARgamma LBD by fluorescence polarization based competitive binding assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College
Curated by ChEMBL
Trinity College
Curated by ChEMBL
Affinity DataEC50: 682nMAssay Description:Agonist activity at PPARgamma LBD in human 293H DA cells after 16 hrs by TR-FRET activation reporter assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College
Curated by ChEMBL
Trinity College
Curated by ChEMBL
Affinity DataEC50: 5.45E+3nMAssay Description:Displacement of pan-PPAR fluormone from PPARgamma LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair