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Found 2 Enz. Inhib. hit(s) with Target = 'Plasmepsin I' and Ligand = 'BDBM50173747'
TargetPlasmepsin I(Plasmodium falciparum)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50173747((1R,2R,3R,4R)-1,4-Bis-((E)-3-bromo-allyloxy)-1,4-b...)
Affinity DataKi:  35nMAssay Description:Inhibition constant against plasmepsin 4 of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50173747((1R,2R,3R,4R)-1,4-Bis-((E)-3-bromo-allyloxy)-1,4-b...)
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition constant against plasmepsin 1 of Plasmodium falciparum, 10 min using 3 uM of DABCYL-Glu-Arg-Nle-Phe-Le u-Ser-Phe-Pro-EDANS as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed