Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50011875'
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Rhone-Poulenc Sante

Curated by PDSP Ki Database
LigandPNGBDBM50011875(2-Bromo-4-(2-chloro-phenyl)-9-methyl-6H-1-thia-5,7...)
Affinity DataKi:  17.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Rhone-Poulenc Sante

Curated by PDSP Ki Database
LigandPNGBDBM50011875(2-Bromo-4-(2-chloro-phenyl)-9-methyl-6H-1-thia-5,7...)
Affinity DataKi:  80.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Rhone-Poulenc Sante

Curated by PDSP Ki Database
LigandPNGBDBM50011875(2-Bromo-4-(2-chloro-phenyl)-9-methyl-6H-1-thia-5,7...)
Affinity DataIC50:  300nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed