Report error Found 4 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily A member 3' and Ligand = 'BDBM50115772'
Affinity DataIC50: 0.0120nMAssay Description:Antagonist activity at human Kv1.3 expressed in CHOK1 cells assessed as inhibition of potassium currents by manual whole-cell patch clamp electrophys...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0230nMAssay Description:Displacement of [125I]-ChTX from mouse Kv1.3 after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.11nMAssay Description:Antagonist activity at Kv1.3 in human whole blood assessed as inhibition of thapsigargin-induced IFN-gamma secretion incubated for 30 prior to thapsi...More data for this Ligand-Target Pair
Affinity DataIC50: 3.76nMAssay Description:Antagonist activity at Kv1.3 in human whole blood assessed as inhibition of thapsigargin-induced IL-2 secretion incubated for 30 prior to thapsigargi...More data for this Ligand-Target Pair
