TargetPresenilin-1(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv)
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of gamma secretase in HEK293 cells expressing APP assessed as reduction in amyloid beta levelsMore data for this Ligand-Target Pair