Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Inhibition of gamma secretase-mediated beta amyloid production in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Inhibition of gamma secretase in APP-transfected CHO cellsMore data for this Ligand-Target Pair