Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM50049512'
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049512(5-Bromo-2-((S)-2,2-dimethyl-6-methylene-cyclohexyl...)
Affinity DataKi:  34nMAssay Description:Binding affinity determined for human Progesterone receptor A isoformMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049512(5-Bromo-2-((S)-2,2-dimethyl-6-methylene-cyclohexyl...)
Affinity DataIC50:  290nMAssay Description:Antagonistic potency to the human progesterone receptor measured in the T-47D alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049512(5-Bromo-2-((S)-2,2-dimethyl-6-methylene-cyclohexyl...)
Affinity DataIC50:  597nMAssay Description:Concentration required to give half-maximal inhibition against human Progesterone receptor B isoform in co-transfected CV-1 cell lines.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049512(5-Bromo-2-((S)-2,2-dimethyl-6-methylene-cyclohexyl...)
Affinity DataEC50:  3.26E+3nMAssay Description:Effective concentration against human Progesterone receptor B isoform expressed in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed