Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.13nMAssay Description:Agonist activity at human PRB expressed in CHO cellsMore data for this Ligand-Target Pair