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Affinity DataIC50: 20nMAssay Description:Inhibition of human PCSK9More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human PCSK9 preincubated for 30 mins followed by EGF(A) addition and measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Inhibition of PCSK9 mediated LDLR degradation in human HepG2 cells assessed as restoration of LDLRMore data for this Ligand-Target Pair
Affinity DataKd: 5.5nMAssay Description:Binding affinity to human PCSK9More data for this Ligand-Target Pair
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