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Found 3 Enz. Inhib. hit(s) with Target = 'Prostaglandin E2 receptor EP1 subtype' and Ligand = 'BDBM50493969'
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493969(CHEMBL2442490)
Affinity DataKi:  530nMAssay Description:Binding affinity to human EP1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493969(CHEMBL2442490)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at human EP1 receptor by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493969(CHEMBL2442490)
Affinity DataIC50:  800nMAssay Description:Antagonist activity at human EP1 receptor by intracellular Ca2+ release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed