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Found 5 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-5' and Ligand = 'BDBM50430966'
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430966(CHEMBL2337849)
Affinity DataKi:  2.43E+3nMAssay Description:Mixed type inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430966(CHEMBL2337849)
Affinity DataKi:  5.03E+3nMAssay Description:Mixed type inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430966(CHEMBL2337849)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of chymotrypsin-like activity of yeast 20S proteasome beta-5 subunit using Suc-LLVY-AMC as substrate measured up to 45 mins by fluorescenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430966(CHEMBL2337849)
Affinity DataIC50:  3.19E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as remaining ac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430966(CHEMBL2337849)
Affinity DataIC50:  7.97E+3nMAssay Description:Inhibition of chymotrypsin-like activity of proteasome beta-5 subunit in HEK293 cells using Suc-LLVY-Glo as substrate incubated for 2 hrs prior to su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed