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Report error Found 3 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-5' and Ligand = 'BDBM50430970'
TargetProteasome subunit beta type-5(Human)
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430970(CHEMBL2337845)
Affinity DataKi:  11nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Human)
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430970(CHEMBL2337845)
Affinity DataIC50:  23nMAssay Description:Inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as remaining ac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Human)
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430970(CHEMBL2337845)
Affinity DataIC50:  472nMAssay Description:Inhibition of chymotrypsin-like activity of proteasome beta-5 subunit in HEK293 cells using Suc-LLVY-Glo as substrate incubated for 2 hrs prior to su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed