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Report error Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50101924'
LigandPNGBDBM50101924(15-benzyl-17-oxo-2-oxa-9,11,15,18-tetraazapentacyc...)
Affinity DataIC50:  2.60nMAssay Description:In vitro inhibitory activity to reduce the human farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ras-CVIMMore data for this Ligand-Target Pair
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LigandPNGBDBM50101924(15-benzyl-17-oxo-2-oxa-9,11,15,18-tetraazapentacyc...)
Affinity DataIC50:  30nMAssay Description:In vitro inhibitory activity to reduce the human geranylgeranyl transferase type I (GGPTase-1)-catalyzed incorporation of 3H GGPP (100 nM) into K-Ras...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed