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Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50189300'
LigandPNGBDBM50189300(CHEMBL3826996)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibition of FTase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50189300(CHEMBL3826996)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed