Found 1 Enz. Inhib. hit(s) with Target = 'Protein-glutamine gamma-glutamyltransferase E' and Ligand = 'BDBM50420474'
TargetProtein-glutamine gamma-glutamyltransferase E(Homo sapiens (Human))
Evotec (Uk)
Curated by ChEMBL
Evotec (Uk)
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of thrombin activated human TG3 by fluorescent transamidation assayMore data for this Ligand-Target Pair