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Found 2 Enz. Inhib. hit(s) with Target = 'Proto-oncogene tyrosine-protein kinase receptor Ret' and Ligand = 'BDBM50565633'
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50565633(CHEMBL4784249)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human GST-tagged RET cytoplasmic domain (658 to 1114 residues) expressed in baculovirus expression system using 5-FAM-EEPLY...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50565633(CHEMBL4784249)
Affinity DataIC50:  63nMAssay Description:Inhibition of recombinant human N-terminal GST-HIS6 fused RET V804M mutant (658 to 1114 residues) expressed in Sf9 insect cells using 5-FAM-EEPLYWSFP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed