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Found
1
Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM24853'
Target
RAC-alpha serine/threonine-protein kinase
(Homo sapiens (Human))
Pfizer
Ligand
BDBM24853
(1-{5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,2-d...)
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Affinity Data
IC50: 4.80nM
pH: 7.5 T: 2°C
Assay Description:
A fluorescence polarization IMAP type assay is used. After a 90 min incubation of reaction mixtures containing enzyme, substrate, and inhibitor, IMAP...
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