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Found 2 Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM50372782'
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372782(CHEMBL402579)
Affinity DataIC50:  69nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372782(CHEMBL402579)
Affinity DataIC50:  221nMAssay Description:Inhibition of Akt1 phosphorylation in human C33a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed