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Found 2 Enz. Inhib. hit(s) with Target = 'Receptor-type tyrosine-protein phosphatase alpha' and Ligand = 'BDBM50326561'
TargetReceptor-type tyrosine-protein phosphatase alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50326561(2-(2,3-dihydro-1H-pyrrolo[3,4-b]quinolin-3-yl)acet...)
Affinity DataIC50:  5.50E+3nMpH: 5.0Assay Description:Inhibition of human cytoplasmic protein tyrosine phosphatase A assessed as change in enzyme activity at pH 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50326561(2-(2,3-dihydro-1H-pyrrolo[3,4-b]quinolin-3-yl)acet...)
Affinity DataIC50:  8.10E+3nMpH: 7.0Assay Description:Inhibition of human cytoplasmic protein tyrosine phosphatase A assessed as change in enzyme activity at pH 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed