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Report error Found 3 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-alpha' and Ligand = 'BDBM50382930'
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine

Curated by ChEMBL
LigandPNGBDBM50382930(CHEMBL115097)
Affinity DataKi:  1.34E+3nMAssay Description:Displacement of [3H]-9-cis retinoic acid from recombinant human RXR-alpha LBD by liquid scintillation counting based competitive ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine

Curated by ChEMBL
LigandPNGBDBM50382930(CHEMBL115097)
Affinity DataKd:  1.35E+3nMAssay Description:Binding affinity to human RXR-alpha by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine

Curated by ChEMBL
LigandPNGBDBM50382930(CHEMBL115097)
Affinity DataKd:  260nMAssay Description:Binding affinity to human RXR-alpha LBD incubated for 2 hrs by tryptophan fluorescence quenching assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed