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Found
1
Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase/endoribonuclease IRE1' and Ligand = 'BDBM602918'
Target
Serine/threonine-protein kinase/endoribonuclease IRE1
(Homo sapiens (Human))
Optikira
US Patent
Ligand
BDBM602918
(1-(4-(8-amino-3-isopropyl-5-(4-(methylamino)cycloh...)
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Affinity Data
IC50: 3nM
Assay Description:
The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...
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Target Info
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Ligand Info
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Details
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