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Report error Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PknB' and Ligand = 'BDBM50421672'
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
William S. Middleton Veterans Hospital

Curated by ChEMBL
LigandPNGBDBM50421672(CHEMBL5316225)
Affinity DataKi:  580nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant PknB (1 to 331 residues) expressed in Escherichia coli BL21-Rosetta cells using GarA and ATP as ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
William S. Middleton Veterans Hospital

Curated by ChEMBL
LigandPNGBDBM50421672(CHEMBL5316225)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant PknB (1 to 331 residues) expressed in Escherichia coli BL21-Rosetta cells using GarA and ATP as ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
William S. Middleton Veterans Hospital

Curated by ChEMBL
LigandPNGBDBM50421672(CHEMBL5316225)
Affinity DataKd:  78nMAssay Description:Binding affinity to Mycobacterium tuberculosis recombinant N-terminal His-tagged PknB (1 to 331 residues) expressed in Escherichia coli DH5alpha cell...More data for this Ligand-Target Pair
In DepthDetails PubMed