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Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase TBK1' and Ligand = 'BDBM50111572'
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Cellzome

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataKd:  79nMAssay Description:Binding affinity to TBK1 in human HEK293/K562/placenta/HepG2 cell lysate mixture incubated for 45 mins by kinobeads based assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Cellzome

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataKd:  251nMAssay Description:Binding affinity to TBK1 in human Ramos cell lysate incubated for 45 mins by kinobeads based assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Cellzome

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataKd:  32nMAssay Description:Binding affinity to phosphorylated TBK1 in calyculin A stimulated human Ramos cell lysate incubated for 45 mins by kinobeads based assayMore data for this Ligand-Target Pair