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Found 3 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50029782'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  9.40nMAssay Description:Ability to inhibit [3H]-(+)-pentazocine binding to guinea pig brain Sigma receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  9.40nMAssay Description:Ability to inhibit [3H]-(+)-pentazocine binding to guinea pig brain Sigma receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  23.3nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed