Found 1 Enz. Inhib. hit(s) with Target = 'Sodium- and chloride-dependent GABA transporter 1' and Ligand = 'BDBM50280958'
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Ludwig-Maximilians-University Munich
Curated by ChEMBL
Ludwig-Maximilians-University Munich
Curated by ChEMBL
Affinity DataIC50: 4.79E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK293 cells assessed as reduction in [3H]GABA uptake preincubated cells with photoirradiated compound for 25 m...More data for this Ligand-Target Pair