Found 13 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50005548'
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
Affinity DataKi: 874nMAssay Description:Inhibition the uptake of tritiated serotonin (5-HT) by the serotonin transporter SERT in rat synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
Affinity DataKi: 874nMAssay Description:Inhibition of serotonin (5-HT) uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Biocon Bristol-Myers Squibb R&D Centre
Curated by ChEMBL
Biocon Bristol-Myers Squibb R&D Centre
Curated by ChEMBL
Affinity DataKi: 874nMAssay Description:Binding affinity to SERT (unknown origin)More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Biocon Bristol-Myers Squibb R&D Centre
Curated by ChEMBL
Biocon Bristol-Myers Squibb R&D Centre
Curated by ChEMBL
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Biocon Bristol-Myers Squibb R&D Centre
Curated by ChEMBL
Biocon Bristol-Myers Squibb R&D Centre
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition of human recombinant SERT expressed in HEK cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Biocon Bristol-Myers Squibb R&D Centre
Curated by ChEMBL
Biocon Bristol-Myers Squibb R&D Centre
Curated by ChEMBL
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Biocon Bristol-Myers Squibb R&D Centre
Curated by ChEMBL
Biocon Bristol-Myers Squibb R&D Centre
Curated by ChEMBL
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
Affinity DataIC50: 830nMAssay Description:Effect on synaptosomal uptake inhibition of 5-hydroxytryptamine (5-HT)More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais
Curated by PDSP Ki Database
Lundbeck Ais
Curated by PDSP Ki Database
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of 5-HT uptake in synaptosomal preparation from rat corpus striatum, using [3H]5-HTMore data for this Ligand-Target Pair