Report error Found 33 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 5' and Ligand = 'BDBM81767'
Affinity DataKi: 0.140nMAssay Description:Inhibition of human sst5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Displacement of [125I]-somatostatin from human SSTR5 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Binding affinity against human sst5 receptor at a dose of 10 uMMore data for this Ligand-Target Pair
Affinity DataKi: 0.398nMAssay Description:Binding affinity towards human Somatostatin receptor type 5 (sst5) using Tyr11-[125I]-SRIF as radioligand was determined in COS cellMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Inhibitory constant against human sst5 receptor at a dose of 10 uMMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibitory constant on human somatostatin receptor 5More data for this Ligand-Target Pair
Affinity DataIC50: 0.860nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor rSSTR5More data for this Ligand-Target Pair
Affinity DataIC50: 0.880nMAssay Description:Inhibition of human SSTR5 by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Displacement of 125I-[LTT]-SRIF-28 from human sst5 receptor in HEK293 cells after 2 hrs by autoradiographyMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST5 receptor expressed in HEK293 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.190nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst5 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0650nMAssay Description:Effective concentration on human somatostatin receptor 5More data for this Ligand-Target Pair
Affinity DataKd: 0.977nMAssay Description:Binding assay at human somatostatin receptor 5 (hsst5) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair