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Report error Found 4 Enz. Inhib. hit(s) with Target = 'Sphingosine 1-phosphate receptor 1' and Ligand = 'BDBM50314401'
TargetSphingosine 1-phosphate receptor 1(Human)
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50314401(2-amino-3-hydroxy-2-((R)-6-octyl-1,2,3,4-tetrahydr...)
Affinity DataEC50:  0.0770nMAssay Description:Agonist activity at human S1P1 receptor assessed as effect on calcium mobilization by Gi dependent whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50314401(2-amino-3-hydroxy-2-((R)-6-octyl-1,2,3,4-tetrahydr...)
Affinity DataEC50:  1.95nMAssay Description:Agonist activity at human S1P1 receptor assessed as effect on calcium mobilization by Gq dependent whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50314401(2-amino-3-hydroxy-2-((R)-6-octyl-1,2,3,4-tetrahydr...)
Affinity DataEC50:  1.95nMAssay Description:Agonist activity at human S1P1 receptor assessed as effect on calcium mobilization by Gq dependent whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Human)
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50314401(2-amino-3-hydroxy-2-((R)-6-octyl-1,2,3,4-tetrahydr...)
Affinity DataEC50:  0.0770nMAssay Description:Agonist activity at human S1P1 receptor assessed as effect on calcium mobilization by Gi dependent whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed