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Found 2 Enz. Inhib. hit(s) with Target = 'Sphingosine 1-phosphate receptor 3' and Ligand = 'BDBM50315562'
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Praecis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50315562((R)-2-amino-2-(4-(4-(biphenyl-4-ylmethoxy)-3-(trif...)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of [33P]sphingosine-1-phosphate from human S1P3 receptor expressed in HEK293T cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Praecis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50315562((R)-2-amino-2-(4-(4-(biphenyl-4-ylmethoxy)-3-(trif...)
Affinity DataEC50: >3.00E+3nMAssay Description:Antagonist activity at human S1P3 receptor expressed in HEK293T cells assessed as inhibition of sphingosine-1-phosphate-induced gamma-[35S]GTP bindin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed