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Report error Found 5 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM242743'
TargetSubstance-P receptor(Human)
Euroscreen

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.21E+4nM ΔG°:  -26.6kJ/molepH: 7.4 T: 25°CAssay Description:The affinity of compounds of the invention for the NK-1 receptor was evaluated in CHO recombinant cells which express the human NK-1 receptor. Membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-P receptor(Human)
Euroscreen

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.21E+4nM ΔG°:  -26.6kJ/molepH: 7.4 T: 25°CAssay Description:The affinity of compounds of the invention for the NK-1 receptor was evaluated in CHO recombinant cells which express the human NK-1 receptor. Membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-P receptor(Human)
Euroscreen

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.21E+4nMAssay Description:The affinity of compounds of the invention for the NK-1 receptor was evaluated in CHO recombinant cells which express the human NK-1 receptor. Membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-P receptor(Human)
Euroscreen

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.21E+4nMAssay Description:The affinity of compounds of the invention for the NK-1 receptor was evaluated in CHO recombinant cells which express the human NK-1 receptor. Membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSubstance-P receptor(Human)
Euroscreen

US Patent
LigandPNGBDBM242743(US10030025, Compound 6 | US10836768, Cpd no 6 | US...)
Affinity DataKi:  2.21E+4nMAssay Description:Human NK-1: The affinity of compounds of the invention for the NK-1 receptor was evaluated in CHO recombinant cells which express the human NK-1 rece...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent