Report error Found 10 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50029885'
Affinity DataKi: 4.20nMAssay Description:Tested for binding affinity towards Tachykinin receptor 1 by using [3H]-SP binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in rat brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Compound was tested for its binding affinity to NK1 receptor in [3H]-SP binding assay on rat brain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 8.70nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in mouse brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against Tachykinin receptor 1 in human IM-9 cells using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in guinea pig brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Compound was tested for its binding affinity to NK1 receptor in [3H]-SP binding assay on human IM9 lymphoblasts cultured cell line.More data for this Ligand-Target Pair
Affinity DataIC50: 4.16E+3nMAssay Description:Inhibition of [3H]-SP binding in rat brain membranesMore data for this Ligand-Target Pair