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Found 3 Enz. Inhib. hit(s) with Target = 'Thyroid hormone receptor beta' and Ligand = 'BDBM50448463'
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50448463(CHEMBL3126367)
Affinity DataIC50:  40nMAssay Description:Displacement of [125I]-Triiodothyronine from human recombinant TRbeta1 ligand binding domain after 2 to 3 hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50448463(CHEMBL3126367)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human recombinant TRbeta1 transfected in human HepG2 cells after 8 to 10 hrs by alkaline phosphatase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50448463(CHEMBL3126367)
Affinity DataEC50:  590nMAssay Description:Agonist activity at human recombinant TRbeta1 transfected in CV-1 cells after 8 to 10 hrs by alkaline phosphatase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed