Report error Found 4 Enz. Inhib. hit(s) with Target = 'Thyrotropin-releasing hormone receptor' and Ligand = 'BDBM50196451'
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]N(1)-Me-His-TRH from TRHR1More data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]N(1)-Me-His-TRH from TRHR2More data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 2.40nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 4.90nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair